PDB Entry - 8U2E

(Status - Released)

Summary information:

Title: Bruton's tyrosine kinase in complex with N-[(2R)-1-[(3R)-3-(methylcarbamoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(3-methylphenyl)-1-oxopropan-2-yl]-1H-indazole-5-carboxamide

PDB DOI: https://doi.org/10.2210/pdb8u2e/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.3c01007

Entry authors: Gajewski, S., Clifton, M.C.

Initial deposition on: 5 September 2023

Initial release on: 31 January 2024

Latest revision on: 6 March 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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