PDB Entry - 9GAX (pdb_00009gax)

(Status - Released)

Summary information:

Title: TEAD1 in complex with a reversible inhibitor N-[(1S)-2-hydroxy-1-(1-methyl-1H-pyrazol-3-yl)ethyl]-2-methyl-8-[4-(trifluoromethyl)phenyl]-2H,8H-pyrazolo[3,4-b]indole-5-carboxamide

PDB DOI: https://doi.org/10.2210/pdb9gax/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.4c01949

Entry authors: Musil, D., Freire, F.

Initial deposition on: 29 July 2024

Initial release on: 22 January 2025

Latest revision on: 9 April 2025

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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