PDB Entry - 9QEK (pdb_00009qek)

(Status - Released)

Summary information:

Title: Structure of Human ROS1 Kinase Domain Harboring the G2032R Solvent-front Mutation in Complex with Zidesamtinib (NVL-520)

PDB DOI: https://doi.org/10.2210/pdb9qek/pdb

Primary publication DOI: https://doi.org/10.1158/1535-7163.MCT-25-0025

Entry authors: Tangpeerachaikul, A., Mente, S., Magrino, J., Gu, F., Horan, J.C., Pelish, H.E.

Initial deposition on: 10 March 2025

Initial release on: 30 April 2025

Latest revision on: 14 May 2025

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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